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Exemestane is a steroidal aromatase inhibitor commonly studied for its role in reducing estrogen levels by irreversibly binding to the aromatase enzyme. It is frequently used in research involving estrogen-dependent processes and hormonal regulation.
Exemestane 20 mg / tab
20 tablets
100 in stock
Aromasin, an effective anti-estrogen medication, plays a crucial role in regulating estrogen levels within the body. By preventing estrogenic side effects, it helps users achieve and maintain a lean, dry appearance, particularly when using aromatizable compounds. This effect is especially important for athletes or bodybuilders preparing for a competition, where achieving a hard physique is essential.
Aromasin works by binding to the aromatase enzyme, which is responsible for converting testosterone and other aromatizable substances into estrogen. Once bound, it deactivates the aromatase enzyme permanently, ensuring no further estrogen production. This irreversible inhibition sets Aromasin apart from other anti-estrogens, as not all anti-estrogen medications provide this level of control. It also eliminates the risk of estrogen rebound, a problem common with non-suicidal aromatase inhibitors like anastrozole and letrozole.
Due to its unique mechanism of action, Aromasin is considered a “suicide inhibitor”—a term that highlights its ability to permanently deactivate the aromatase enzyme. While it requires more frequent dosing (twice daily, ideally every 12 hours) to maintain consistent blood levels, this contrasts with other aromatase inhibitors that can be dosed less frequently. Aromasin also stands out for its neutral impact on cholesterol levels, unlike other anti-estrogens that may negatively affect lipid profiles, making it a more heart-friendly option.
Key Benefits:
Permanent inhibition of aromatase enzyme: By binding to aromatase, Aromasin deactivates it, preventing the conversion of testosterone into estrogen.
No estrogen rebound: Unlike non-suicidal inhibitors, Aromasin eliminates the risk of estrogen surge after discontinuation.
Supports heart health: Its steroidal nature avoids the lipid-impacting effects that are common with other aromatase inhibitors.
Enhances testosterone bioavailability: By lowering SHBG (sex hormone-binding globulin), Aromasin improves the effectiveness of testosterone in the body, especially during cycles.
Aids post-cycle therapy (PCT): Aromasin is highly effective for restoring hormonal balance after anabolic steroid cycles.
Testosterone boosting: Studies show a 60% increase in total testosterone and over 100% increase in free testosterone with a 25mg daily dose in just 10 days.
Treatment for gynecomastia: Aromasin has proven effective in reducing symptoms of gynecomastia.
No estrogen rebound: It remains a reliable choice for both on-cycle estrogen control and post-cycle therapy.
Dosage and Administration:
Typical dose: 25mg daily for best results.
Long-acting effect: A single 25mg dose maintains low estrogen levels for up to 72 hours.
Half-life: Approximately 9 hours, ensuring consistent and stable estrogen control.